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Pharmaceutical CI-1033 Canertinib CAS 267243-28-7

Product Detail Information

 

 

 

 

 


Product Name: Canertinib
Synonyms: N-[4-(3-chloro-4-fluoroanilino)-7-(3-morpholin-4-ylpropoxy)quinazolin-6-yl]prop-2-enamide;N-[4-(3-chloro-4-fluoro-anilino)-7-(3-morpholinopropoxy)quinazolin-6-yl]acrylamide;CI-1033(Canertinib);PD-183805;Canertinib base;Canetinib;Canertinib (CI-1033);N-[4-(3-chloro-4-fluoroanilino)-7-(3-Morpholin-4-ylpropoxy)quinazolin-6-yl]prop-2-en
CAS: 267243-28-7
MF: C24H25ClFN5O3
MW: 485.944
EINECS:  
Product Categories: Inhibitors
Mol File: 267243-28-7.mol

 

 


Usage:
1.Antineoplastic; irreversible pan-erbB tyrosine kinase inhibitor used to treat cancer. 
2.CI-1033 is a potent inhibitor of EGFR and ErbB2 with IC50 of 1.5 nM and 9.0 nM, respectively. 

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